SEP-4199
SEP4199 is an orally active 5-HT7 receptor ligand, with a Ki value of 66 nM for human 5-HT7R and 16 nM for human D2R. SEP4199 mediates antidepressant effects. SEP4199 is applicable for the research of bipolar depression.
For research use only. We do not sell to patients.
- CAS No.: 2974362-88-2
- Formula: C17H27N3O4S
- Molecular Weight:369.48
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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D2 Receptor 16 nM (Ki) |
5-HT7 Receptor 66 nM (Ki) |
SEP4199 exhibits a higher relative affinity for human recombinant 5-HT7 receptors than human recombinant D2 receptors, with a 5-HT7R Ki of 66 ± 16 nM and a D2R Ki of 16 ± 0.62 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2974362-88-2
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Molecular Weight 369.48
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Formula C17H27N3O4S
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SMILES
CCN1[C@@H](CNC(C2=CC(S(=O)(CC)=O)=C(N)C=C2OC)=O)CCC1.CCN3[C@H](CNC(C4=CC(S(=O)(CC)=O)=C(N)C=C4OC)=O)CCC3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
SEP-4199 Related Classifications
HY-14545B Related Classifications
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