JYL-273
JYL-273 is a TRPV1 agonist, with the IC50 of 361 nM in CHO-TRPV1 cell lines.
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- CAS 番号: 1391826-17-7
- 分子式: C28H39NO4S
- 分子量:485.68
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
361 nM (CHO-TRPV1 cell lines)[1].
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CHO | EC50 |
1.34 nM
Compound: 2
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Agonist activity at human TRPV1 expressed in CHO cells assessed as 45Ca2+ uptake after 20 mins by liquid scintillation counting analysis
Agonist activity at human TRPV1 expressed in CHO cells assessed as 45Ca2+ uptake after 20 mins by liquid scintillation counting analysis
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[PMID: 24321344] |
| CHO | EC50 |
2.83 nM
Compound: 2
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In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cells
In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cells
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[PMID: 12825950] |
化学情報
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CAS 番号 1391826-17-7
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分子量 485.68
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分子式 C28H39NO4S
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SMILES
CC(C)(C)C(OCC(CC1=CC=C(C(C)(C)C)C=C1)CC(NCC2=CC=C(O)C(OC)=C2)=S)=O
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
JYL-273 関連分類
HY-128479 関連分類
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