JYL-79
JYL-79 is a TRPV1 agonist with the IC50 of 3.9 nM. JYL-79 can be used for study of neuropathic pain.
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 289902-64-3
- 分子式: C26H36N2O4S
- 分子量:472.64
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| CHO | EC50 |
1.97 nM
Compound: 1
|
In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cells
In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cells
|
[PMID: 12825950] |
| CHO | EC50 |
1.97 nM
Compound: 2
|
Agonist activity at rat TRPV1 expressed in CHO cells assessed as maximal calcium uptake
Agonist activity at rat TRPV1 expressed in CHO cells assessed as maximal calcium uptake
|
[PMID: 17035013] |
化学情報
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CAS 番号 289902-64-3
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分子量 472.64
-
分子式 C26H36N2O4S
-
SMILES
CC(C)(C)C(OCC(CNC(NCC1=CC=C(O)C(OC)=C1)=S)CC2=CC=C(C)C(C)=C2)=O
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輸送条件
Room temperature in continental US; may vary elsewhere.
-
保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)