LSD1/HDAC6-IN-1
LSD1/HDAC6-IN-1 is an orally active dual inhibitor of lysine specific demethylase 1(LSD1)/Histone deacetylase 6 (HDAC6), with anti-tumor activity. LSD1/HDAC6-IN-1 can be used for the research of multiple myeloma (MM).
For research use only. We do not sell to patients.
- CAS No.: 2738306-38-0
- Formula: C25H33N3O2
- Molecular Weight:407.55
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
Biological Activity
|
KDM1/LSD1 |
HDAC6 |
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| RPMI-8226 | EC50 |
0.28 μM
Compound: 1
|
Antiproliferative activity against human RPMI-8226 cells assessed as reduction in cell viability after 144 hrs
Antiproliferative activity against human RPMI-8226 cells assessed as reduction in cell viability after 144 hrs
|
[PMID: 33359604] |
LSD1/HDAC6-IN-1 shows superior potency in multiple MM lines[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
CAS No. 2738306-38-0
-
Molecular Weight 407.55
-
Formula C25H33N3O2
-
SMILES
ONC(C(C=C1)=CC=C1CCCN(CC2)CCC2CN[C@@H]3[C@@H](C4=CC=CC=C4)C3)=O
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
LSD1/HDAC6-IN-1 Related Classifications
HY-131970 Related Classifications
Powered by Bioz