NPD13668
NPD13668 is an EZH2-mediated gene silencing modulator. NPD13668 inhibits EZH2/PRC2 (polycomb repressive complex 2) activity. NPD13668 reactivates the expression of silenced H3K27me3 target genes together with depletion of the H3K27me3 modification. NPD13668 can be used for the study of prostate cancer and ovarian cancer.
For research use only. We do not sell to patients.
- CAS No.: 864819-54-5
- Formula: C22H20N2O5
- Molecular Weight:392.40
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Histone Methyltransferase Isoforms
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Biological Activity
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EZH2 |
Chemical Information
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CAS No. 864819-54-5
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Molecular Weight 392.40
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Formula C22H20N2O5
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SMILES
O=C(NCCC1=CNC2=C1C=CC=C2)CC3=C(C)C4=CC=C(O)C(O)=C4OC3=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)