PROTAC BRD2 BD1 Degrader-1
PROTAC BRD2 BD1 Degrader-1 (compound 21-1) is a potent and selective BRD2 BD1 PROTAC degrader. PROTAC BRD2 BD1 Degrader-1 induces the association of BRD2 BD1 and von Hippel–Lindau-elongin C-elongin B (VCB).
(Pink: BRD2 BD1 ligand (HY-175679); Blue: VHL ligand (HY-125845); Black: linker).
For research use only. We do not sell to patients.
- Formula: C51H66N12O4S
- Molecular Weight:943.21
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All PROTACs Isoforms
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Biological Activity
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BRD2 BD1 |
Chemical Information
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Molecular Weight 943.21
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Formula C51H66N12O4S
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SMILES
CC1=CC=CC2=C1CCN(C2)C3=NC(N4CCC(CC4)CCC(N[C@@H](C(C)(C)C)C(N5C[C@@H](C[C@H]5C(NCC6=CC=C(C=C6)C7=C(N=CS7)C)=O)O)=O)=O)=NC(N8CCC(C8)C9=NC=CN9C)=N3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)