1. Epigenetics
    TGF-beta/Smad
  2. PKC

PKC-theta inhibitor 

Cat. No.: HY-112681
Handling Instructions

PKC-theta inhibitor is a selective PKC-θinhibitor, with an IC50 of 12 nM.

For research use only. We do not sell to patients.

PKC-theta inhibitor Chemical Structure

PKC-theta inhibitor Chemical Structure

CAS No. : 736048-65-0

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  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

PKC-theta inhibitor is a selective PKC-θinhibitor, with an IC50 of 12 nM.

IC50 & Target

PKCθ

12 nM (IC50)

Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.2005 mL 11.0023 mL 22.0046 mL
5 mM 0.4401 mL 2.2005 mL 4.4009 mL
10 mM 0.2200 mL 1.1002 mL 2.2005 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

454.45

Formula

C₂₀H₂₅F₃N₆O₃

CAS No.

736048-65-0

SMILES

FC(F)(F)OC1=CC=CC=C1CNC2=NC=C([N+]([O-])=O)C(NCC3CCC(CN)CC3)=N2

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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This equation is commonly abbreviated as: C1V1 = C2V2

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× = ×
C1   V1   C2   V2

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Product Name:
PKC-theta inhibitor
Cat. No.:
HY-112681
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PKC-theta inhibitor

Cat. No.: HY-112681