1. GPCR/G Protein
    Neuronal Signaling
  2. 5-HT Receptor
    Dopamine Receptor
  3. Brexpiprazole D8

Brexpiprazole D8 (Synonyms: OPC-34712 D8)

Cat. No.: HY-15780S
Handling Instructions

Brexpiprazole D8 (OPC-34712 D8) is a deuterium labeled Brexpiprazole (OPC-34712). Brexpiprazole, an atypical antipsychotic drug, is a partial agonist of human 5-HT1A and dopamine receptor (Ki=0.12 nM and 0.3 nM, respectively). Brexpiprazole is also a 5-HT2A receptor antagonist (Ki=0.47 nM).

For research use only. We do not sell to patients.

Brexpiprazole D8 Chemical Structure

Brexpiprazole D8 Chemical Structure

CAS No. : 1427049-21-5

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Description

Brexpiprazole D8 (OPC-34712 D8) is a deuterium labeled Brexpiprazole (OPC-34712). Brexpiprazole, an atypical antipsychotic drug, is a partial agonist of human 5-HT1A and dopamine receptor (Ki=0.12 nM and 0.3 nM, respectively). Brexpiprazole is also a 5-HT2A receptor antagonist (Ki=0.47 nM)[1][2].

Molecular Weight

441.62

Formula

C₂₅H₁₉D₈N₃O₂S

CAS No.

1427049-21-5

SMILES

O=C1NC2=C(C=CC(OCCCCN3C([2H])([2H])C([2H])([2H])N(C4=C(C=CS5)C5=CC=C4)C([2H])([2H])C3([2H])[2H])=C2)C=C1

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Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

Brexpiprazole D8OPC-34712 D8Brexpiprazole D 8Brexpiprazole D-85-HT ReceptorDopamine ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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