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  3. CBP/p300-IN-2

CBP/EP300-IN-2 is an inhibitor of CBP/EP300 with IC50 values of 1.07 nM and 5.96 nM for CBP/HTRF and Myc, respectively. CBP/EP300-IN-2, example 25, is extracted from patent WO2017205538A1.

For research use only. We do not sell to patients.

CBP/p300-IN-2 Chemical Structure

CBP/p300-IN-2 Chemical Structure

CAS No. : 2158265-96-2

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Description

CBP/EP300-IN-2 is an inhibitor of CBP/EP300 with IC50 values of 1.07 nM and 5.96 nM for CBP/HTRF and Myc, respectively. CBP/EP300-IN-2, example 25, is extracted from patent WO2017205538A1[1].

IC50 & Target

IC50:1.07 nM (CBP/HTRF); 5.96 nM (Myc)[1]

Molecular Weight

521.56

Formula

C27H29F2N7O2

CAS No.
SMILES

O=C(N1CCC(N(C2CCOCC2)N=C3C4=CN=CC5=C4C=C(C(F)F)C(C6=CN(C)N=C6)=C5)=C3C1)NC

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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CBP/p300-IN-2 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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CBP/p300-IN-2
Cat. No.:
HY-128761
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