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CBP/EP300-IN-2 

Cat. No.: HY-128761
Handling Instructions

CBP/EP300-IN-2 is an inhibitor of CBP/EP300 with IC50 values of 0.00107 μM and 0.00596 μM for CBP/HTRF and Myc, respectively. CBP/EP300-IN-2, example 25, is extracted from patent WO2017205538A1.

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CBP/EP300-IN-2 Chemical Structure

CBP/EP300-IN-2 Chemical Structure

CAS No. : 2158265-96-2

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Description

CBP/EP300-IN-2 is an inhibitor of CBP/EP300 with IC50 values of 0.00107 μM and 0.00596 μM for CBP/HTRF and Myc, respectively. CBP/EP300-IN-2, example 25, is extracted from patent WO2017205538A1[1].

IC50 & Target

IC50: 0.00107 μM (CBP/HTRF); 0.00596 μM (Myc)[1]

Molecular Weight

521.56

Formula

C₂₇H₂₉F₂N₇O₂

CAS No.

2158265-96-2

SMILES

O=C(N1CCC(N(C2CCOCC2)N=C3C4=CN=CC5=C4C=C(C(F)F)C(C6=CN(C)N=C6)=C5)=C3C1)NC

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Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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CBP/EP300-IN-2
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