1. Neuronal Signaling
    GPCR/G Protein
    Metabolic Enzyme/Protease
  2. Dopamine Receptor
    5-HT Receptor
    Drug Metabolite
  3. Desmethyl cariprazine

Desmethyl cariprazine 

Cat. No.: HY-100656
Handling Instructions

Desmethyl cariprazine is an active metabolite of Cariprazine. Cariprazine, an antipsychotic drug candidate, exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM).

For research use only. We do not sell to patients.

Desmethyl cariprazine Chemical Structure

Desmethyl cariprazine Chemical Structure

CAS No. : 839712-15-1

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Description

Desmethyl cariprazine is an active metabolite of Cariprazine[1]. Cariprazine, an antipsychotic drug candidate, exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM)[2].

Molecular Weight

413.38

Formula

C₂₀H₃₀Cl₂N₄O

CAS No.

839712-15-1

SMILES

O=C(NC)N[[email protected]@H]1CC[[email protected]@H](CCN2CCN(C3=CC=CC(Cl)=C3Cl)CC2)CC1

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

Desmethyl cariprazineDopamine Receptor5-HT ReceptorDrug MetaboliteSerotonin Receptor5-hydroxytryptamine ReceptoractivemetaboliteantipsychotictolerabilityInhibitorinhibitorinhibit

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Desmethyl cariprazine
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