CDK2 modulator 1
CDK2 modulator 1 is a CDK2 modulator with an EC50 < 100 nM and an Emax > 100% of positive control in a TR-FRET proximity assay. CDK2 modulator 1 induces ternary complex formation with CDK2/CCNE1 and CRBN. CDK2 modulator 1 can be used for the research of cancer.
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 3066623-95-5
- 分子式: C30H27FN6O5
- 分子量:570.57
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
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CDK2/cyclinE |
CDK2 modulator 1 (compound 248) (10-point dilution series; 2 h (room temperature)) induces ternary complex formation between purified CDK2/CCNE1 and CRBN/DDB1 proteins with an EC50 < 100 nMl[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 3066623-95-5
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分子量 570.57
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分子式 C30H27FN6O5
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SMILES
N#CC1=CC(C2=CC(OC)=C(C(C)(C)NC(NC3=CC=C4C(N(C5C(NC(CC5)=O)=O)CC4=C3F)=O)=O)C=C2)=CN=C1
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
CDK2 modulator 1 関連分類
HY-186126 関連分類
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