DC-CPin711
Based on 1 Customer Validation
DC-CPin711 is a potent and selective inhibitor of CREB-binding protein (CBP) bromodomain with an IC50 of 0.0626 μM. DC-CPin711 arrests cell cycle at G1 phase and induces apoptosis.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度: 99.09%
- CAS 番号: 2447559-21-7
- 分子式: C23H22N4O2
- 分子量:386.45
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保管条件:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
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Apoptosis Compound Library
HY-L003
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Epigenetics Compound Library
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Histone Modification Research Compound Library
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Anti-Cancer Compound Library
HY-L025
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Reprogramming Compound Library
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Anti-Blood Cancer Compound Library
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Anti-Obesity Compound Library
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Transcription Factor-Targeted Library
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Anti-Prostate Cancer Compound Library
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Anti-Pulmonary Fibrosis Compound Library
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Heterocyclic Compound Library
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Pain-Related Compound Library
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Highly Selective Inhibitors Library
HY-L158
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Highly Selective Activators Library
HY-L159
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Cell Death Library
HY-L162
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Anti-Hematopathy Compound Library
HY-L171
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Bioactive Compound Library Max
HY-L181
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MCE Bioactive Compound Library
HY-L001V
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Bioactive Compound Library
HY-L001
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Non-Alcoholic Fatty Liver Disease (NAFLD) Compound Library
HY-L199
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High-Throughput Bioactive Compound Library
HY-L205
生物活性
IC50: 0.0626 μM (CBP bromodomain)[1]
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CWR22R | IC50 |
13 μM
Compound: 17
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Antiproliferative activity against human 22RV-1 cells incubated for 96 hrs by CellTiter-Glo luminescent assay
Antiproliferative activity against human 22RV-1 cells incubated for 96 hrs by CellTiter-Glo luminescent assay
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[PMID: 33045661] |
| MV4-11 | IC50 |
1.2 μM
Compound: 17
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Antiproliferative activity against human MV4-11 cells incubated for 96 hrs by CellTiter-Glo luminescent assay
Antiproliferative activity against human MV4-11 cells incubated for 96 hrs by CellTiter-Glo luminescent assay
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[PMID: 33045661] |
化学情報
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CAS 番号 2447559-21-7
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性状 Solid
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分子量 386.45
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分子式 C23H22N4O2
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Color white
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SMILES
O=C(N1CCCC2=C1C=C(NC(C3=CC=CC(C4=CC=NC=C4)=C3)=O)C=C2)NC
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
純度とドキュメンテーション
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データシート (266 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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取扱説明書 (2659 KB)
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
DC-CPin711 関連分類
HY-147868 関連分類
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