Milsaperidone
Milsaperidone ((S)-Hydroxy Iloperidone; VHX-896) is an orally active serotonin 5-HT2A and dopamine D2 receptor antagonist. Milsaperidone ((S)-Hydroxy Iloperidone) is the active metabolite of the antipsychotic agent Iloperidone (HY-17410). Milsaperidone can be used in studies related to mental disorders such as depression.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 501373-88-2
- 分子式: C24H29FN2O4
- 分子量:428.50
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性
製品説明
体内実験
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
臨床実験
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | 2011-05 | PHASE1 |
化学情報
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CAS 番号 501373-88-2
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分子量 428.50
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分子式 C24H29FN2O4
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SMILES
FC1=CC=C(C(C2CCN(CC2)CCCOC3=C(C=C(C=C3)[C@@H](O)C)OC)=NO4)C4=C1
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別名
(S)-Hydroxy Iloperidone; VHX-896
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
Keywords
- Milsaperidone
- 501373-88-2
- (S)-Hydroxy Iloperidone
- VHX-896
- VHX896
- VHX 896
- VHX-896
- Drug Metabolite
- Dopamine Receptor
- 5-HT Receptor
- somnolence
- acute bipolar I disorder
- major depressive disorder
- iloperidone
- QTc prolongation
- schizophrenia
- serotonin 5-HT2A receptor
- dopamine D2 receptor
- weight gain
- Inhibitor
- inhibitor
- inhibit