Mefuparib
Based on 1 Customer Validation
Mefuparib (CVL218) is a poly ADP-ribose polymerase (PARP) inhibitor used in cancer research that exhibits potent brain penetration due to its high protein binding.
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- Purity: 99.77%
- CAS No.: 1392502-82-7
- 화학식: C17H15FN2O2
- 분자량:298.31
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보관:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
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용액&용해도
- 순도&문서
- References
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Help & FAQs
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Cell Cycle/DNA Damage Compound Library
HY-L004
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Epigenetics Compound Library
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Anti-Cancer Compound Library
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Clinical Compound Library
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HY-L034
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Anti-Pancreatic Cancer Compound Library
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Anti-Ovarian Cancer Compound Library
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Bioactive Compound Library Max
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HY-L035P
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Clinical Compound Library Plus
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Bioactive Compound Library
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Biological Activity
| NCT Number | Sponsor | Condition | Start Date |
Phase
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|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 1392502-82-7
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Appearance Solid
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분자량 298.31
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화학식 C17H15FN2O2
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Color White to off-white
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SMILES
O=C(C1=CC(F)=CC2=C1OC(C3=CC=C(CNC)C=C3)=C2)N
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Synonyms
CVL218
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
용액&용해도
DMSO : 6.25 mg/mL (20.95 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
순도&문서
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Data Sheet (267 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 3.3522 mL | 16.7611 mL | 33.5222 mL | 83.8054 mL |
| 5 mM | 0.6704 mL | 3.3522 mL | 6.7044 mL | 16.7611 mL | |
| 10 mM | 0.3352 mL | 1.6761 mL | 3.3522 mL | 8.3805 mL | |
| 15 mM | 0.2235 mL | 1.1174 mL | 2.2348 mL | 5.5870 mL | |
| 20 mM | 0.1676 mL | 0.8381 mL | 1.6761 mL | 4.1903 mL |
Mefuparib Related Classifications
HY-167927 Related Classifications
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