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MMSET-IN-1 

Cat. No.: HY-124699
Handling Instructions

MMSET-IN-1 is a multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) inhibitor against SETD2 and MMSET with IC50s of 0.49 and 3.3 μM, respectively. MMSET-IN-1 has a Kd of 1.6 μM for MMSET.

For research use only. We do not sell to patients.

MMSET-IN-1 Chemical Structure

MMSET-IN-1 Chemical Structure

CAS No. : 1998139-29-9

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Description

MMSET-IN-1 is a multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) inhibitor against SETD2 and MMSET with IC50s of 0.49 and 3.3 μM, respectively. MMSET-IN-1 has a Kd of 1.6 μM for MMSET[1].

IC50 & Target

IC50: 0.49 μM (SETD2), 3.3 μM (MMSET)[1]
Kd: 1.6 μM[1]

Molecular Weight

423.47

Formula

C₁₈H₂₉N₇O₅

CAS No.

1998139-29-9

SMILES

O=C(O)[[email protected]@H](N)CCC(NCCC)C[[email protected]]1O[[email protected]@H](N2C=NC3=C(N)N=CN=C23)[[email protected]](O)[[email protected]@H]1O

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Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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