PARP1-IN-53
PARP1-IN-53 (Compound 328) is a quinazolinone derivative and PARP1 inhibitor with a PARP1 IC50 of 0.1 nM and selectivity over PARP2, which has a PARP2 IC50 of 23 nM.PARP1-IN-53 can be used for the research of cancer.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- CAS. Nr.: 3087853-45-7
- Formel: C22H19N5O3
- Molecular Weight:401.42
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
Beschreibung
IC50 & Target
[1]|
PARP-1 0.1 nM (IC50) |
PARP-2 23 nM (IC50) |
Chemical Information
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CAS. Nr. 3087853-45-7
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Molecular Weight 401.42
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Formel C22H19N5O3
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SMILES
O=C1NC(/C=C/C(N2CCN(C3=CC=C(C#N)C=C3)CC2)=O)=NC4=C(O)C=CC=C41
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)