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Referencia número: HY-181332

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PROTAC EZH2 Degrader-37

PROTAC EZH2 Degrader-37 (compound 16) is a PROTAC protein degrader targeting EZH2 with a target IC₅₀ of 144 nM. PROTAC EZH2 Degrader-37 is applicable to lymphoma-related research.
(Pink: EZH2 ligand (HY-147230); Blue: Cereblon ligand (HY-103596); Black: linker).

Para uso exclusivo en investigación. No vendemos a pacientes.

No. CAS: 2653338-73-7
Fòrmula: C₅₇H₇₃N₇O₈
Peso molecular:984.23

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

PROTAC EZH2 Degrader-37 Chemical Structure

No. CAS: 2653338-73-7

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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- In Vitro
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Actividad biológica

Descripciòn

PROTAC EZH2 Degrader-37 (compound 16) is a PROTAC protein degrader targeting EZH2 with a target IC₅₀ of 144 nM. PROTAC EZH2 Degrader-37 is applicable to lymphoma-related research^[1]. (Pink: EZH2 ligand (HY-147230); Blue: Cereblon ligand (HY-103596); Black: linker).

Ver todos los productos específicos de isoformas PROTACs :

Ver todos los productos específicos de isoformas Histone Methyltransferase :

In Vitro

PROTAC EZH2 Degrader-37 (compound 16) inhibits EZH2 enzymatic activity with an IC₅₀ of 144.00 nM^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .

Chemical Information

No. CAS 2653338-73-7
Peso molecular 984.23
Fòrmula C₅₇H₇₃N₇O₈
SMILES

CCN(C1CCOCC1)C2=CC(C3=CC=C(C=C3)CN4CCN(CC4)CCCCCCCCCCOC5=C(C6=CC=C5)C(N(C6=O)C7CCC(NC7=O)=O)=O)=CC(C(NCC8=C(C=C(NC8=O)C)C)=O)=C2C
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureza y Documentación

Instrucciones de manejo (2659 KB)

Referencias

[1]. S Abulkhair H, et al. Therapeutic horizons in the development of PROTAC-based EZH2 inhibitors: recent achievements, comparative analysis, and future perspectives. RSC Adv. 2026;16(4):3034-3056. Published 2026 Jan 14. [Content Brief]

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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PROTAC EZH2 Degrader-37

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PROTAC EZH2 Degrader-37

Ver todos los productos específicos de isoformas PROTACs

Ver todos los productos específicos de isoformas Histone Methyltransferase

Actividad biológica

Descripciòn

In Vitro

Chemical Information

Pureza y Documentación

Referencias

Calculators

Help & FAQs

PROTAC EZH2 Degrader-37 Related Classifications

HY-181332 Related Classifications

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