2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. TRP Channel
  4. ABT-102

ABT-102 is a potent and highly selective Vanilloid Receptor (TRPV1) receptor antagonist. ABT-102 potently and reversibly increases heat pain thresholds and reduced painfulness of suprathreshold oral/cutaneous heat. ABT-102 reduces nociceptive responses of animals in models of inflammatory, bone cancer, postoperative, and osteoarthritic pain.

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ABT-102 Chemical Structure

ABT-102 Chemical Structure

CAS No. : 808756-71-0

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Based on 1 publication(s) in Google Scholar

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Description

ABT-102 is a potent and highly selective Vanilloid Receptor (TRPV1) receptor antagonist. ABT-102 potently and reversibly increases heat pain thresholds and reduced painfulness of suprathreshold oral/cutaneous heat. ABT-102 reduces nociceptive responses of animals in models of inflammatory, bone cancer, postoperative, and osteoarthritic pain[1][2].

IC50 & Target

TRPV1

 

Molecular Weight

348.44

Formula

C21H24N4O
CAS No.
SMILES

O=C(NC1=CC=CC2=C1C=NN2)N[C@@H]3CCC4=C3C=CC(C(C)(C)C)=C4
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Room temperature in continental US; may vary elsewhere.
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Purity & Documentation
References
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ABT-102 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

ABT-102808756-71-0ABT102ABT 102TRP ChannelTransient receptor potential channelsInhibitorinhibitorinhibit

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