2. Epigenetics
  3. Histone Methyltransferase
  4. DCPT1061

DCPT1061 potently inhibits PRMT1, PRMT6 and PRMT8 in vitro with less inhibitory effect on PRMT3, PRMT4, and PRMT5 or other epigenetic enzymes. DCPT1061 has antitumor effect.

For research use only. We do not sell to patients.

DCPT1061 Chemical Structure

DCPT1061 Chemical Structure

CAS No. : 2289726-31-2

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5 mg USD 225 In-stock
10 mg USD 360 In-stock
25 mg USD 720 In-stock
50 mg USD 1150 In-stock
100 mg USD 1800 In-stock
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Based on 1 publication(s) in Google Scholar

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Description

DCPT1061 potently inhibits PRMT1, PRMT6 and PRMT8 in vitro with less inhibitory effect on PRMT3, PRMT4, and PRMT5 or other epigenetic enzymes. DCPT1061 has antitumor effect[1][2].

Molecular Weight

339.26

Formula

C17H20Cl2N2O
CAS No.
Appearance

Liquid

Color

Colorless to light yellow

SMILES

ClC1=C(OC2=CC=CC=C2CN(C)CCNC)C=CC=C1Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Solvent & Solubility
In Vitro: 

DMSO : ≥ 250 mg/mL (736.90 mM; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.9476 mL 14.7380 mL 29.4759 mL
5 mM 0.5895 mL 2.9476 mL 5.8952 mL
View the Complete Stock Solution Preparation Table

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  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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In Vivo Dissolution Calculator
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Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.9476 mL 14.7380 mL 29.4759 mL 73.6898 mL
5 mM 0.5895 mL 2.9476 mL 5.8952 mL 14.7380 mL
10 mM 0.2948 mL 1.4738 mL 2.9476 mL 7.3690 mL
15 mM 0.1965 mL 0.9825 mL 1.9651 mL 4.9127 mL
20 mM 0.1474 mL 0.7369 mL 1.4738 mL 3.6845 mL
25 mM 0.1179 mL 0.5895 mL 1.1790 mL 2.9476 mL
30 mM 0.0983 mL 0.4913 mL 0.9825 mL 2.4563 mL
40 mM 0.0737 mL 0.3684 mL 0.7369 mL 1.8422 mL
50 mM 0.0590 mL 0.2948 mL 0.5895 mL 1.4738 mL
60 mM 0.0491 mL 0.2456 mL 0.4913 mL 1.2282 mL
80 mM 0.0368 mL 0.1842 mL 0.3684 mL 0.9211 mL
100 mM 0.0295 mL 0.1474 mL 0.2948 mL 0.7369 mL
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DCPT1061 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

DCPT10612289726-31-2DCPT 1061DCPT-1061Histone MethyltransferaseInhibitorinhibitorinhibit

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