1. Epigenetics
  2. Histone Methyltransferase
  3. EZH2-​IN-​2

EZH2-​IN-​2 

Cat. No.: HY-A0298
Handling Instructions

EZH2-IN-2 is a EZH2 inhibitor extracted from patent WO2018133795A1, Compound Example 69, with an IC50 of 64 nM. EZH2-IN-2 can be used for the research of cancer or precancerous condition related to EZH2 activity.

For research use only. We do not sell to patients.

EZH2-​IN-​2 Chemical Structure

EZH2-​IN-​2 Chemical Structure

CAS No. : 2238821-31-1

Size Price Stock Quantity
10 mM * 1  mL in DMSO USD 5644 In-stock
Estimated Time of Arrival: December 31
1 mg USD 200 In-stock
Estimated Time of Arrival: December 31
5 mg USD 420 In-stock
Estimated Time of Arrival: December 31
10 mg USD 700 In-stock
Estimated Time of Arrival: December 31
50 mg USD 2000 Get quote
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200 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

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Description

EZH2-IN-2 is a EZH2 inhibitor extracted from patent WO2018133795A1, Compound Example 69, with an IC50 of 64 nM. EZH2-IN-2 can be used for the research of cancer or precancerous condition related to EZH2 activity[1].

IC50 & Target[1]

EZH2

64 nM (IC50)

Molecular Weight

610.79

Formula

C₃₆H₄₆N₆O₃

CAS No.

2238821-31-1

SMILES

O=C(NCC1=C(C)C=C(C)NC1=O)C2=CC(C3=CC=C(N4CCN(CC5CC5)CC4)N=C3C)=CC(N(C(C6CC6)=O)CC)=C2C

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

EZH2-​IN-​2Histone MethyltransferaseEZH2histonemethyltransferaseInhibitorinhibitorinhibit

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EZH2-​IN-​2
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