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  3. PROTAC BET degrader-3

PROTAC BET degrader-3 

Cat. No.: HY-114229 Purity: 98.64%
Handling Instructions

PROTAC BET Degrader-3 is a potent BET degrader based on PROTAC.

For research use only. We do not sell to patients.

PROTAC BET degrader-3 Chemical Structure

PROTAC BET degrader-3 Chemical Structure

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 977 In-stock
Estimated Time of Arrival: December 31
5 mg USD 550 In-stock
Estimated Time of Arrival: December 31
10 mg USD 850 In-stock
Estimated Time of Arrival: December 31
25 mg USD 1850 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
100 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

PROTAC BET Degrader-3 is a potent BET degrader based on PROTAC.

IC50 & Target

BET[1]

Molecular Weight

1045.22

Formula

C₅₃H₆₄N₁₂O₉S

SMILES

CCN1N=C(C2CC2)C=C1NC3=NC(C(NCCOCCOCC(N[[email protected]@H](C(C)(C)C)C(N4[[email protected]](C(NCC5=CC=C(C6=C(C)N=CS6)C=C5)=O)C[[email protected]@H](O)C4)=O)=O)=O)=NC7=C3C8=CC(OC)=C(C(C(C)=NO9)=C9C)C=C8N7

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -20°C 3 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (95.67 mM; Need ultrasonic)

H2O : < 0.1 mg/mL (insoluble)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 0.9567 mL 4.7837 mL 9.5674 mL
5 mM 0.1913 mL 0.9567 mL 1.9135 mL
10 mM 0.0957 mL 0.4784 mL 0.9567 mL
*Please refer to the solubility information to select the appropriate solvent.
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  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
PROTAC BET degrader-3
Cat. No.:
HY-114229
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