Pimethixene
Pimethixene is antihistamine and antiserotonergic compound, acts as an antimigraine agent. Pimethixene is a highly potent antagonist of 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors, with pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively.
For research use only. We do not sell to patients.
- CAS No.: 314-03-4
- Formula: C19H19NS
- Molecular Weight:293.43
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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5-HT1A Receptor |
5-HT2A Receptor |
5-HT2B Receptor |
5-HT2C Receptor |
5-HT2B Receptor 10.44 (pKi) |
5-HT2A Receptor 10.22 (pKi) |
5-HT2C Receptor 8.42 (pKi) |
5-HT1A Receptor 7.63 (pKi) |
M2 receptor 9.38 (pKi) |
M1 receptor 8.61 (pKi) |
D2 receptor 8.19 (pKi) |
DD4.4 receptor 7.54 (pKi) |
Chemical Information
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CAS No. 314-03-4
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Molecular Weight 293.43
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Formula C19H19NS
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SMILES
CN1CC/C(CC1)=C2C3=C(SC4=C\2C=CC=C4)C=CC=C3
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Synonyms
Pimetixene
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pimethixene Related Classifications
HY-B1101 Related Classifications
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