Pimethixene
Pimethixene is antihistamine and antiserotonergic compound, acts as an antimigraine agent. Pimethixene is a highly potent antagonist of 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors, with pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively.
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- No. CAS: 314-03-4
- Fòrmula: C19H19NS
- Peso molecular:293.43
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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Chemical Information
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Ver todos los productos específicos de isoformas 5-HT Receptor
MoreVer todos los productos específicos de isoformas Histamine Receptor
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Actividad biológica
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5-HT1A Receptor |
5-HT2A Receptor |
5-HT2B Receptor |
5-HT2C Receptor |
5-HT2B Receptor 10.44 (pKi) |
5-HT2A Receptor 10.22 (pKi) |
5-HT2C Receptor 8.42 (pKi) |
5-HT1A Receptor 7.63 (pKi) |
M2 receptor 9.38 (pKi) |
M1 receptor 8.61 (pKi) |
D2 receptor 8.19 (pKi) |
DD4.4 receptor 7.54 (pKi) |
Chemical Information
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No. CAS 314-03-4
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Peso molecular 293.43
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Fòrmula C19H19NS
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SMILES
CN1CC/C(CC1)=C2C3=C(SC4=C\2C=CC=C4)C=CC=C3
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Synonyms
Pimetixene
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pimethixene Related Classifications
HY-B1101 Related Classifications
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