HDAC1-IN-3
HDAC1-IN-3 is a potent Pf HDAC1 inhibitor. HDAC1-IN-3 shows antimalarial activity in wild-type and multidrug-resistant parasite strains. HDAC1-IN-3 shows a significant in vivo killing effect against all life cycles of parasites.
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 2482998-35-4
- 分子式: C22H24ClN7O2
- 分子量:453.92
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
Parasite アイソフォーム固有の製品をすべて表示
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生物活性
製品説明
IC50 & Target
|
HDAC1 2.2 nM (IC50) |
HDAC2 5.1 nM (IC50) |
HDAC3 5.2 nM (IC50) |
HDAC6 85.5 nM (IC50) |
HDAC8 29.9 nM (IC50) |
Plasmodium |
Cellular Effect
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| HEK-293T | IC50 |
1.21 μM
Compound: JX35
|
Cytotoxicity against HEK293T cells incubated for 72 hrs by CCK-8 assay
Cytotoxicity against HEK293T cells incubated for 72 hrs by CCK-8 assay
|
[PMID: 35175762] |
| HepG2 | IC50 |
1.02 μM
Compound: JX35
|
Cytotoxicity against human HepG2 cells incubated for 72 hrs by CCK-8 assay
Cytotoxicity against human HepG2 cells incubated for 72 hrs by CCK-8 assay
|
[PMID: 35175762] |
体外実験
HDAC1-IN-3 (compound JX35) shows antimalarial activity with IC50s of 1.26 nM and 1.61 nM for wild-type Plasmodium falciparum (P. falciparum) parasite 3D7 and chloroquine-resistant P. falciparum parasite Dd2, respectively[1].
HDAC1-IN-3 (10 µM; 72 h) shows low cytotoxicity with IC50s of 1.02 µM and 1.21 µM for HepG2, 293T cells, respectively[1].
HDAC1-IN-3 (72 h) shows no cross-resistance with clinical antimalarial drugs with IC50s of 3.06, 2.18, 5.85 nM for GB4, C2A, CP286, respectively[1].
HDAC1-IN-3 (10, 30, 60, 100 nM; 3, 6, 12, 24 h) shows antimalarial activity in a time- and dose-dependent manner with asynchronous 3D7 parasites[1].
HDAC1-IN-3 (40 nM, 4 days; P. falciparum 3D7 cells) shows the killing effects of JX35 on P. falciparum parasites during asexual reproduction stages might be related to the inhibition of schizont growth and reinvasion of RBCs (red blood cells)[1].
HDAC1-IN-3 (5, 20 nM; 4 h) inhibits the expression of Pf HDAC against ART (artemisinin)-resistant parasite strains[1].
HDAC1-IN-3 reduces the inhibition of hHDACs with IC50s of 2.2, 5.1, 5.2, 85.5, 29.9 nM for HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
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Cell Line:HepG2, 293T cells
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Concentration:10 µM
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Incubation Time:72 h
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Result:Showed low cytotoxicity with IC50s of 1.02 µM and 1.21 µM for HepG2, 293T cells, respectively.
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Cell Line:P. falciparum 3D7 cells
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Concentration:5, 20 nM
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Incubation Time:4 h
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Result:Inhibited the expression of Pf HDAC against ART (artemisinin)-resistant parasite strains.
体内実験
HDAC1-IN-3 (5 mg/kg; i.p.) shows good pharmacokinetic properties[1].
Pharmacokinetic Parameters of HDAC1-IN-3 in Female BALB/c mice[1].
| parameter | JX35 |
| Cmax (ng/mL) | 539 |
| Tmax (h) | 0.25 |
| AUC last (h·ng/mL) | 638 |
| AUC inf (h·ng/mL) | 640 |
| t1/2 (h) | 0.91 |
| CLZ/F (L/h/kg) | 7.81 |
| VZ/F (L/kg) | 10.20 |
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
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Animal Model:6-8 weeks, BALB/c female mice[1]
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Dosage:30, 60, 90 mg/kg
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Administration:I.p., once daily for 5 days
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Result:Showed acceptable therapeutic efficacy and safety.
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Animal Model:6-8 weeks, female BALB/c mice[1]
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Dosage:5 mg/kg
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Administration:I.p.
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Result:Showed good pharmacokinetic properties.
化学情報
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CAS 番号 2482998-35-4
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分子量 453.92
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分子式 C22H24ClN7O2
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SMILES
O=C(C1=CN=C(N(CC2)CC32CN(CC4=CN(C)C5=C4C=CC(C#N)=C5)C3)N=C1)NO.[H]Cl
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)