PQR530 (Standard)
PQR530 (Standard) is the analytical standard of PQR530 (HY-107365). This product is intended for research and analytical applications. PQR530 is a potent, ATP-competitive, orally bioavailable and brain-penetrant dual pan-PI3K/mTORC1/2 inhibitor, with a subnanomolar Kd toward PI3Kα and mTOR (0.84 and 0.33 nM, respectively). Antitumor activity.
For research use only. We do not sell to patients.
- CAS No.: 1927857-61-1
- Formula: C18H23F2N7O2
- Molecular Weight:407.42
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
PI3K/mTORC1/2[1]
Chemical Information
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CAS No. 1927857-61-1
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Molecular Weight 407.42
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Formula C18H23F2N7O2
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SMILES
FC(C1=CC(N)=NC=C1C2=NC(N3CCOCC3)=NC(N4[C@H](COCC4)C)=N2)F
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)