1. Epigenetics
  2. Histone Methyltransferase
  3. SETD2-IN-1 TFA

SETD2-IN-1 TFA 

Cat. No.: HY-136328
Handling Instructions

SETD2-IN-1 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase. SETD2-IN-1 TFA has anti-proliferative effects.

For research use only. We do not sell to patients.

SETD2-IN-1 TFA Chemical Structure

SETD2-IN-1 TFA Chemical Structure

CAS No. : 2411759-92-5

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Description

SETD2-IN-1 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase. SETD2-IN-1 TFA has anti-proliferative effects[1].

IC50 & Target

SETD2[1]

Molecular Weight

514.51

Formula

C₂₄H₃₀F₄N₄O₄

CAS No.

2411759-92-5

SMILES

O=C(C(N1)=CC2=C1C(C)=CC=C2F)N[[email protected]]3C[[email protected]@H](N4CCN(C(C)=O)CC4)CCC3.O=C(O)C(F)(F)F

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

SETD2-IN-1Histone MethyltransferasecancerSETD2histonemethyltransferasesInhibitorinhibitorinhibit

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SETD2-IN-1 TFA
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