1. GPCR/G Protein
    Neuronal Signaling
  2. Opioid Receptor

Trimebutine maleate 

Cat. No.: HY-B0380A Purity: 99.95%
Handling Instructions

Trimebutine maleate is a drug with antimuscarinic and weak mu opioid agonist effects.

For research use only. We do not sell to patients.

Trimebutine maleate Chemical Structure

Trimebutine maleate Chemical Structure

CAS No. : 34140-59-5

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply now  
10 mM * 1 mL in DMSO USD 66 In-stock
Stock in Sweden
Estimated Time of Arrival: December 31
5 g USD 60 In-stock
Stock in Sweden
Estimated Time of Arrival: December 31
10 g   Get quote  
50 g   Get quote  

* Please select Quantity before adding items.

Other Forms of Trimebutine maleate:

  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

Trimebutine maleate is a drug with antimuscarinic and weak mu opioid agonist effects. Target: Opioid Receptor Trimebutine is an agonist of peripheral mu, kappa and delta opiate receptors, used as spasmolytic agent for treatment of both acute and chronic abdominal pain [1]. The major product from drug metabolism of trimebutine in human beings is nor-trimebutine, which comes from removal of one of the methyl groups attached to nitrogen. Trimebutine exerts its effects in part due to causing a premature activation of phase III of the migrating motor complex in the digestive tract [2, 3].

Clinical Trial
Solvent & Solubility
In Vitro: 

DMSO : ≥ 38 mg/mL (75.47 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.9859 mL 9.9297 mL 19.8594 mL
5 mM 0.3972 mL 1.9859 mL 3.9719 mL
10 mM 0.1986 mL 0.9930 mL 1.9859 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

503.54

Formula

C₂₆H₃₃NO₉

CAS No.

34140-59-5

SMILES

O=C(O)/C=C\C(O)=O.O=C(OCC(C1=CC=CC=C1)(N(C)C)CC)C2=CC(OC)=C(OC)C(OC)=C2

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Inquiry Online

Your information is safe with us. * Required Fields.

Product name

 

Salutation

Applicant name *

 

Email address *

Phone number *

 

Organization name *

Country or Region *

 

Requested quantity *

Remarks

Bulk Inquiry

Inquiry Information

Product Name:
Trimebutine maleate
Cat. No.:
HY-B0380A
Quantity:

Trimebutine maleate

Cat. No.: HY-B0380A