BL-1020 mesylate
BL-1020 mesylate is the mesylate salt form of BL-1020. BL-1020 mesylate is an antipsychotic agent. BL-1020 mesylate is inhibitor for dopamine receptor and serotonin receptor (5-HT receptor), with Ki of 0.066, 0.062 and 0.21 nM, for D2L, D2S and 5-HT2A receptors, respectively. BL-1020 mesylate is agonist for GABAA receptor with Ki of 3.74 μM, and enhances the GABA release. BL-1020 mesylate exhibits high affinity with histamine receptor (Ki is 0.47 nM). BL-1020 mesylate reduces Amphetamine-induced hyperactivity, with lower catalepsy and sedation. BL-1020 mesylate is blood-brain barrier penetrate.
For research use only. We do not sell to patients.
- CAS No.: 916898-61-8
- Formula: C26H37ClN4O5S2
- Molecular Weight:585.18
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All 5-HT Receptor Isoforms
MoreAll Dopamine Receptor Isoforms
MoreAll Histamine Receptor Isoforms
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Biological Activity
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5-HT2A Receptor |
D2S Receptor 0.062 nM (Ki) |
D2L Receptor 0.066 nM (Ki) |
Histamine Receptor 0.47 nM (Ki) |
5-HT2A Receptor 3.74 μM (Ki) |
Chemical Information
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CAS No. 916898-61-8
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Molecular Weight 585.18
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Formula C26H37ClN4O5S2
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SMILES
O=C(CCCN)OCCN1CCN(CCCN2C3=C(SC4=CC=C(C=C42)Cl)C=CC=C3)CC1.O=S(O)(C)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
BL-1020 mesylate Related Classifications
HY-111136 Related Classifications
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