1. Metabolic Enzyme/Protease
  2. Phospholipase
  3. GSK2647544

GSK2647544 

Cat. No.: HY-145653
Handling Instructions

GSK2647544 is an orally available, selective inhibitor of Lp-PLA2. Lipoprotein-associated phospholipase (Lp-PLA2) is a calcium-independent phospholipase A2 with proinflammatory activities that is primarily secreted by monocyte-derived macrophages.

For research use only. We do not sell to patients.

GSK2647544 Chemical Structure

GSK2647544 Chemical Structure

CAS No. : 1380426-95-8

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Description

GSK2647544 is an orally available, selective inhibitor of Lp-PLA2. Lipoprotein-associated phospholipase (Lp-PLA2) is a calcium-independent phospholipase A2 with proinflammatory activities that is primarily secreted by monocyte-derived macrophages[1].

Molecular Weight

502.87

Formula

C24H18ClF3N4O3

CAS No.
SMILES

O=C1NC(OCCC2=CC=C(C=C2)OC3=CC=C(C(C(F)(F)F)=C3)Cl)=NC=C1CC4=CN=CN=C4

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
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GSK2647544
Cat. No.:
HY-145653
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