1. Membrane Transporter/Ion Channel
    Neuronal Signaling
    Metabolic Enzyme/Protease
  2. TRP Channel
    Endogenous Metabolite
  3. OMDM-5

OMDM-5 

Cat. No.: HY-135881
Handling Instructions

OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU), with a Ki of 4.8 μM. OMDM-5 is also a potent vanilloid receptor type 1 (VR1, TRPV1) agonist, with an EC50 of 75 nM, and shows weakly active as cannabinoid receptor type 1 (CB1) ligand (Ki=4.9 μM).

For research use only. We do not sell to patients.

OMDM-5 Chemical Structure

OMDM-5 Chemical Structure

CAS No. : 616884-66-3

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Description

OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU), with a Ki of 4.8 μM. OMDM-5 is also a potent vanilloid receptor type 1 (VR1, TRPV1) agonist, with an EC50 of 75 nM, and shows weakly active as cannabinoid receptor type 1 (CB1) ligand (Ki=4.9 μM)[1].

IC50 & Target

Ki: 4.8 μM (anandamide cellular uptake), 4.9 μM (CB1), EC50: 75 nM (VR1)[1]

Molecular Weight

432.64

Formula

C₂₆H₄₄N₂O₃

CAS No.

616884-66-3

SMILES

CCCCCCCC/C=C\CCCCCCCC(NNCC1=CC=C(O)C(OC)=C1)=O

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

OMDM-5OMDM5OMDM 5TRP ChannelEndogenous MetaboliteTransient receptor potential channelsfattyacidsuptakeRBL-2H3cellsvanilloidVR1cannabinoidreceptortype1CB1CB2FAAHInhibitorinhibitorinhibit

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OMDM-5
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