2. Cell Cycle/DNA Damage Epigenetics
  3. PARP
  4. PARP7-IN-16

PARP7-IN-16 (compound 36) is a potent, selective and orally active inhibitor of PARP-1/2/7, with IC50s of 0.94, 0.87 and 0.21 nM, respectively. PARP7-IN-16 can be used for the research of breast cancer and prostate cancer.

For research use only. We do not sell to patients.

PARP7-IN-16 Chemical Structure

PARP7-IN-16 Chemical Structure

CAS No. : 2435657-10-4

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PARP7-IN-16 Related Antibodies

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Description

PARP7-IN-16 (compound 36) is a potent, selective and orally active inhibitor of PARP-1/2/7, with IC50s of 0.94, 0.87 and 0.21 nM, respectively. PARP7-IN-16 can be used for the research of breast cancer and prostate cancer[1].

IC50 & Target[1]

PARP-1

0.94 nM (IC50)

PARP-2

0.87 nM (IC50)

PARP-7

0.21 nM (IC50)

Molecular Weight

488.49

Formula

C25H26FN4NaO4
CAS No.
SMILES

O=C([N-]C1=O)C2=CC=CC=C2N1CC3=CC=C(C(C(N4CCN(C(C4)=O)C(CC)CC)=O)=C3)F.[Na+]
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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PARP7-IN-16 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PARP7-IN-162435657-10-4PARPpoly ADP ribose polymerasebreast cancerprostate cancerInhibitorinhibitorinhibit

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