1. GPCR/G Protein
    Neuronal Signaling
  2. 5-HT Receptor
    Dopamine Receptor
  3. Pipamperone

Pipamperone (Synonyms: Floropipamide; McN-JR 3345; R 3345)

Cat. No.: HY-100703 Purity: 99.89%
Handling Instructions

Pipamperone (Floropipamide; McN-JR 3345; R 3345) is a high-affinity antagonist of 5-HT2A receptor (pKi=8.2) and D4 receptor (pKi=8.0) and a low-affinity antagonist of D2 receptor (pKi=6.7).

For research use only. We do not sell to patients.

Pipamperone Chemical Structure

Pipamperone Chemical Structure

CAS No. : 1893-33-0

Size Price Stock Quantity
10 mM * 1 mL in Water USD 165 In-stock
Estimated Time of Arrival: December 31
5 mg USD 150 In-stock
Estimated Time of Arrival: December 31
10 mg   Get quote  
50 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

Pipamperone (Floropipamide; McN-JR 3345; R 3345) is a high-affinity antagonist of 5-HT2A receptor (pKi=8.2) and D4 receptor (pKi=8.0) and a low-affinity antagonist of D2 receptor (pKi=6.7)[1].

IC50 & Target[1]

5-HT2A Receptor

8.2 (pKi)

5-HT2C Receptor

6.9 (pKi)

5-HT1 Receptor

5.7 (pKi)

D4 receptor

8.0 (pKi)

D2 receptor

6.7 (pKi)

α1 receptor

7.2 (pKi)

Clinical Trial
Molecular Weight

375.48

Formula

C₂₁H₃₀FN₃O₂

CAS No.

1893-33-0

SMILES

O=C(C1(N2CCCCC2)CCN(CCCC(C3=CC=C(F)C=C3)=O)CC1)N

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, protect from light, stored under argon

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light, stored under argon)

Solvent & Solubility
In Vitro: 

0.1 M HCL : 25 mg/mL (66.58 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.6633 mL 13.3163 mL 26.6326 mL
5 mM 0.5327 mL 2.6633 mL 5.3265 mL
10 mM 0.2663 mL 1.3316 mL 2.6633 mL
*Please refer to the solubility information to select the appropriate solvent.
References

Purity: 99.89%

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KeyWords:

Pipamperone | Floropipamide | McN-JR 3345 | R 3345 | R3345 | R 3345 | R-3345 | 5-HT Receptor | Dopamine Receptor | Serotonin Receptor | 5-hydroxytryptamine Receptor | Inhibitor | inhibitor | inhibit

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Pipamperone
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HY-100703
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