PROTAC BRD4 Degrader-29
PROTAC BRD4 Degrader-29 (compound 7a) is a potent PROTACs degrader of BRD4, with the DC50 of 89.4 nM. PROTAC BRD4 Degrader-29 plays an important role in cancer research (Pink: ligand for target protein (HY-13030); Black: linker (HY-172125); Blue: E3 ligase ligand (HY-103597)).
(Pink: BRD4 ligand (HY-13030); Blue: Cereblon ligand (HY-103597); Black: linker (HY-172125)).
For research use only. We do not sell to patients.
- Formula: C58H61ClN10O9S2
- Molecular Weight:1141.75
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All PROTACs Isoforms
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Biological Activity
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BRD4 89.4 nM (DC50) |
Chemical Information
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Molecular Weight 1141.75
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Formula C58H61ClN10O9S2
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SMILES
CC1=NN=C2N1C3=C(C(C4=CC=C(Cl)C=C4)=N[C@H]2CC(NCCNC(C5=CC=C(SCCC#CC(C6CCOCC6)N7CCC(NC(COC8=CC=CC9=C8C(N(C%10CCC(NC%10=O)=O)C9=O)=O)=O)CC7)C=C5)=O)=O)C(C)=C(C)S3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)