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  3. BPKDi

BPKDi 

Cat. No.: HY-118052
Handling Instructions

BPKDi is a potent bipyridyl PKD inhibitor with IC50s of 1 nM, 9 nM and 1 nM for PKD1, PKD2 and PKD3, respectively. BPKDi blocks signal-dependent phosphorylation and nuclear export of class IIa HDACs in cardiomyocytes.

For research use only. We do not sell to patients.

BPKDi Chemical Structure

BPKDi Chemical Structure

CAS No. : 1201673-28-0

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Description

BPKDi is a potent bipyridyl PKD inhibitor with IC50s of 1 nM, 9 nM and 1 nM for PKD1, PKD2 and PKD3, respectively. BPKDi blocks signal-dependent phosphorylation and nuclear export of class IIa HDACs in cardiomyocytes[1].

IC50 & Target[1]

PKD1

1 nM (IC50)

PKD2

9 nM (IC50)

PKD3

1 nM (IC50)

Molecular Weight

380.49

Formula

C21H28N6O

CAS No.
SMILES

O=C(N)C1=CC(C2=CC(NC3CCCCC3)=NC=C2)=NC(N4CCNCC4)=C1

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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BPKDi
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HY-118052
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