CCT68127
CCT68127 is an orally active CDK inhibitor. CCT68127 can be used in anti-cancer research.
Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.
- CAS No.: 660822-23-1
- Formule: C19H27N7O
- Masse moléculaire:369.46
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
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CDK2 |
CDK7 |
CDK9 |
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HT-29 | IC50 |
1.3 μM
Compound: alphaSbetaR-21, CCT68127
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Inhibition of CDK7 in human HT29 cells assessed as reduction in RNA polymerase 2 expression
Inhibition of CDK7 in human HT29 cells assessed as reduction in RNA polymerase 2 expression
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[PMID: 21982796] |
| HT-29 | IC50 |
107 nM
Compound: alphaSbetaR-21, CCT68127
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Inhibition of CDK9 in human HT29 cells assessed as reduction in RNA polymerase 2 expression
Inhibition of CDK9 in human HT29 cells assessed as reduction in RNA polymerase 2 expression
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[PMID: 21982796] |
Chemical Information
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CAS No. 660822-23-1
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Masse moléculaire 369.46
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Formule C19H27N7O
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SMILES
C[C@@H](O)[C@@H](NC1=NC(NCC2=CC=CN=C2)=C3N=CN(C(C)C)C3=N1)CC
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Synonyms
αSβR-21
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CCT68127 Related Classifications
HY-123826 Related Classifications
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