1. Cell Cycle/DNA Damage
  2. CDK
  3. CDK2-IN-4

CDK2-IN-4 

Cat. No.: HY-117535
Handling Instructions

CDK2-IN-4 is a potent and selective CDK2 inhibitor with an IC50 of 44 nM for CDK2/cyclin A, shows 2,000-fold selectivity over CDK1/cyclin B (IC50=86 uM).

For research use only. We do not sell to patients.

CDK2-IN-4 Chemical Structure

CDK2-IN-4 Chemical Structure

CAS No. : 2079895-42-2

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Description

CDK2-IN-4 is a potent and selective CDK2 inhibitor with an IC50 of 44 nM for CDK2/cyclin A, shows 2,000-fold selectivity over CDK1/cyclin B (IC50=86 uM)[1].

IC50 & Target[1]

cdk2/cyclin A

44 nM (IC50)

Cdk1/cyclin B

86 μM (IC50)

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Molecular Weight

442.49

Formula

C₂₃H₁₈N₆O₂S

CAS No.

2079895-42-2

SMILES

O=S(C1=CC=C(C=C1)NC2=NC3=NC=NC3=C(C4=CC(C5=CC=CC=C5)=CC=C4)N2)(N)=O

Shipping

Room temperature in continental US; may vary elsewhere

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

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× = ×
C1   V1   C2   V2

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CDK2-IN-4
Cat. No.:
HY-117535
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CDK2-IN-4

Cat. No.: HY-117535