HL403
HL403 is a potent and dual BRD4/Src inhibitor. HL403 has IC50 values of 133 nM for BRD4 inhibition and 4.5 nM for Src inhibition. HL403 shows anti-cancer activity.
For research use only. We do not sell to patients.
- Formula: C44H46Cl2N12O4S2
- Molecular Weight:941.95
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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BRD4 133 nM (IC50) |
Chemical Information
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Molecular Weight 941.95
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Formula C44H46Cl2N12O4S2
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SMILES
CC1=C(C)SC2=C1C(C3=CC=C(C=C3)Cl)=N[C@H](C4=NN=C(N42)C)CC(N[C@@H](C)C(OCCN5CCN(CC5)C6=NC(C)=NC(NC7=NC=C(S7)C(NC8=C(C=CC=C8Cl)C)=O)=C6)=O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)