CCT68127
CCT68127 is an orally active CDK inhibitor. CCT68127 can be used in anti-cancer research.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 660822-23-1
- 分子式: C19H27N7O
- 分子量:369.46
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
|
CDK2 |
CDK7 |
CDK9 |
|
Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HT-29 | IC50 |
1.3 μM
Compound: alphaSbetaR-21, CCT68127
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Inhibition of CDK7 in human HT29 cells assessed as reduction in RNA polymerase 2 expression
Inhibition of CDK7 in human HT29 cells assessed as reduction in RNA polymerase 2 expression
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[PMID: 21982796] |
| HT-29 | IC50 |
107 nM
Compound: alphaSbetaR-21, CCT68127
|
Inhibition of CDK9 in human HT29 cells assessed as reduction in RNA polymerase 2 expression
Inhibition of CDK9 in human HT29 cells assessed as reduction in RNA polymerase 2 expression
|
[PMID: 21982796] |
化学情報
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CAS 番号 660822-23-1
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分子量 369.46
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分子式 C19H27N7O
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SMILES
C[C@@H](O)[C@@H](NC1=NC(NCC2=CC=CN=C2)=C3N=CN(C(C)C)C3=N1)CC
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別名
αSβR-21
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
CCT68127 関連分類
HY-123826 関連分類
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