1. Cell Cycle/DNA Damage
  2. CDK

BGG463 

Cat. No.: HY-100600 Purity: >98.0%
Handling Instructions

BGG463 is a CDK2 inhibitor.

For research use only. We do not sell to patients.

BGG463 Chemical Structure

BGG463 Chemical Structure

CAS No. : 890129-26-7

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 318 In-stock
Estimated Time of Arrival: December 31
5 mg USD 250 In-stock
Estimated Time of Arrival: December 31
10 mg USD 350 In-stock
Estimated Time of Arrival: December 31
25 mg USD 750 In-stock
Estimated Time of Arrival: December 31
50 mg USD 1200 In-stock
Estimated Time of Arrival: December 31
100 mg USD 1900 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

BGG463 is a CDK2 inhibitor.

IC50 & Target[1]

CDK2

 

Solvent & Solubility
In Vitro: 

DMSO : ≥ 125 mg/mL (216.05 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.7284 mL 8.6418 mL 17.2837 mL
5 mM 0.3457 mL 1.7284 mL 3.4567 mL
10 mM 0.1728 mL 0.8642 mL 1.7284 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.08 mg/mL (3.60 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.08 mg/mL (3.60 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.08 mg/mL (3.60 mM); Clear solution

References
Molecular Weight

578.58

Formula

C₃₀H₂₉F₃N₆O₃

CAS No.

890129-26-7

SMILES

O=C(C1=C2C=CC(OC3=NC=NC(NC(C)=O)=C3)=CC2=CC=C1)NC4=CC=C(CN5CCN(C)CC5)C(C(F)(F)F)=C4

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Inquiry Information

Product Name:
BGG463
Cat. No.:
HY-100600
Quantity:

BGG463

Cat. No.: HY-100600