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DFCI-002-06

DFCI-002-06 is an orally active dual-target HCK/BTK PROTAC degrader with DC₅₀ values for HCK and BTK of 1.3 and 4.5 nM respectively. DFCI-002-06 retains higher anti-tumor activity than the HCK/BTK dual-target inhibitor (HY-15805), inducing apoptosis in cancer cells. DFCI-002-06 can be used for the study of MYD88 mutant B-cell malignancies.
(Pink: Src and Btk ligand (HY-15805); Blue: Cereblon ligand (HY-W087383); Black: linker).

商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。

  • CAS 番号: 3092208-36-8
  • 分子式: C44H46N10O5
  • 分子量:794.90
  • 保管条件:

    Please store the product under the recommended conditions in the Certificate of Analysis.

  • DFCI-002-06 Chemical Structure
    DFCI-002-06 構造式
CAS 番号: 3092208-36-8
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  • DFCI-002-06 Chemical Structure
    DFCI-002-06 Chemical Structure
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  • DFCI-002-06