CDK2 modulator 1
CDK2 modulator 1 is a CDK2 modulator with an EC50 < 100 nM and an Emax > 100% of positive control in a TR-FRET proximity assay. CDK2 modulator 1 induces ternary complex formation with CDK2/CCNE1 and CRBN. CDK2 modulator 1 can be used for the research of cancer.
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- No. CAS: 3066623-95-5
- Fòrmula: C30H27FN6O5
- Peso molecular:570.57
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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CDK2/cyclinE |
CDK2 modulator 1 (compound 248) (10-point dilution series; 2 h (room temperature)) induces ternary complex formation between purified CDK2/CCNE1 and CRBN/DDB1 proteins with an EC50 < 100 nMl[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 3066623-95-5
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Peso molecular 570.57
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Fòrmula C30H27FN6O5
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SMILES
N#CC1=CC(C2=CC(OC)=C(C(C)(C)NC(NC3=CC=C4C(N(C5C(NC(CC5)=O)=O)CC4=C3F)=O)=O)C=C2)=CN=C1
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CDK2 modulator 1 Related Classifications
HY-186126 Related Classifications
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