1. PROTAC
    Epigenetics
  2. PROTAC
    Epigenetic Reader Domain
  3. VZ185

VZ185 

Cat. No.: HY-114322
Handling Instructions

VZ185 is a potent, fast, and selective dual BRD7/9 PROTAC degrader with DC50s of 4.5 and 1.8 nM, respectively.

For research use only. We do not sell to patients.

VZ185 Chemical Structure

VZ185 Chemical Structure

CAS No. : 2306193-61-1

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Description

VZ185 is a potent, fast, and selective dual BRD7/9 PROTAC degrader with DC50s of 4.5 and 1.8 nM, respectively.

IC50 & Target

DC50: 4.5 nM (BRD7), 1.8 nM (BRD9)[1]

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Molecular Weight

995.21

Formula

C₅₃H₆₇FN₈O₈S

CAS No.

2306193-61-1

SMILES

O=C([[email protected]]1N(C([[email protected]@H](NC(C2(F)CC2)=O)C(C)(C)C)=O)C[[email protected]](O)C1)NCC3=CC=C(C4=C(C)N=CS4)C=C3OCCCCCN5CCN(CC6=C(OC)C=C(C(C7=CC=NC=C87)=CN(C)C8=O)C=C6OC)CC5

Shipping

Room temperature in continental US; may vary elsewhere

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
VZ185
Cat. No.:
HY-114322
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VZ185

Cat. No.: HY-114322