Rac-Pemafibrate
Pemafibrate racemate (K13675 racemate) is the racemate of pemafibrate, and activates PPARα activity, with EC50s of 1 nM, >10 μM and 1.7 μM for h-PPARα, h-PPARγ and h-PPARδ, respectively.
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- CAS No.: 848258-31-1
- Formule: C28H30N2O6
- Masse moléculaire:490.55
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
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h-PPARα 1 nM (EC50) |
h-PPARδ 1.7 μM (EC50) |
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 848258-31-1
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Masse moléculaire 490.55
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Formule C28H30N2O6
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SMILES
CCC(OC1=CC=CC(CN(C2=NC3=CC=CC=C3O2)CCCOC4=CC=C(OC)C=C4)=C1)C(O)=O
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Synonyms
Rac-K13675
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)