Antitrypanosomal agent 31
Antitrypanosomal agent 31 is an antitrypanosoma agent with a pEC50 of 6.4. Antitrypanosomal agent 31 inhibits GSK-3β, CDK-2, and CDK-4 with pIC50s of 5.8, 6.9, and 7.1, respectively. Antitrypanosomal agent 31 can be used for the research of human african trypanosomiasis.
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- CAS. Nr.: 551919-54-1
- Formel: C13H12N6
- Molecular Weight:252.28
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
Beschreibung
IC50 & Target
[1]|
Trypanosoma 6.4 (pEC50) |
human CDK2 6.9 (pIC50) |
human CDK4 7.1 (pIC50) |
GSK-3β 5.8 (pIC50) |
In Vitro
Antitrypanosomal agent 31 (Compound 10c) inhibits Trypanosoma brucei growth with a pEC50 of 6.4, while also inhibiting human CDK-2, CDK-4, and GSK-3β kinases with pIC50s of 5.8, 6.9, and 7.1, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS. Nr. 551919-54-1
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Molecular Weight 252.28
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Formel C13H12N6
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SMILES
N1=CC=C(N=C1NC2CC2)C=3C=NN4N=CC=CC34
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
Antitrypanosomal agent 31 Related Classifications
HY-183529 Related Classifications
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