Antitrypanosomal agent 31
Antitrypanosomal agent 31 is an antitrypanosoma agent with a pEC50 of 6.4. Antitrypanosomal agent 31 inhibits GSK-3β, CDK-2, and CDK-4 with pIC50s of 5.8, 6.9, and 7.1, respectively. Antitrypanosomal agent 31 can be used for the research of human african trypanosomiasis.
For research use only. We do not sell to patients.
- CAS No.: 551919-54-1
- Formula: C13H12N6
- Molecular Weight:252.28
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Biological Activity
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Trypanosoma 6.4 (pEC50) |
human CDK2 6.9 (pIC50) |
human CDK4 7.1 (pIC50) |
GSK-3β 5.8 (pIC50) |
Antitrypanosomal agent 31 (Compound 10c) inhibits Trypanosoma brucei growth with a pEC50 of 6.4, while also inhibiting human CDK-2, CDK-4, and GSK-3β kinases with pIC50s of 5.8, 6.9, and 7.1, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 551919-54-1
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Molecular Weight 252.28
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Formula C13H12N6
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SMILES
N1=CC=C(N=C1NC2CC2)C=3C=NN4N=CC=CC34
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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