CDK8/BRD4-IN-1
CDK8/BRD4-IN-1 is a dual CDK8/BRD4 inhibitor, with an IC50 of 5.44 μM against CDK8 and an IC50 of 4.03 μM against BRD4. CDK8/BRD4-IN-1 exhibits anticancer activity against colorectal cancer. CDK8/BRD4-IN-1 can be used for the research of colorectal cancer.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- Formel: C27H36N6O
- Molecular Weight:460.61
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
Beschreibung
IC50 & Target
[1]|
CDK8 5.44 μM (IC50) |
BRD4 4.03 μM (IC50) |
In Vitro
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Molecular Weight 460.61
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Formel C27H36N6O
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SMILES
CN(C(C=C1)=C(N(C(C)C)[C@@H]2C)C=C1NCCCCCCNC3=NC=NC4=C3C=CC=C4)C2=O
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)