CDK9/PARP-IN-1
CDK9/PARP-IN-1 (compound 37) is a CDK9/PARP inhibitor. CDK9/PARP-IN-1 inhibits CDK9 and PARP1 with IC50s of 118 and 107 nM, respectively. CDK9/PARP-IN-1 exhibits broad-spectrum antiproliferative effects across multiple cancer cell lines.
For research use only. We do not sell to patients.
- CAS No.: 3032818-67-7
- Formula: C38H34F2N8O3
- Molecular Weight:688.73
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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CDK9 118 nM (IC50) |
PARP1 107 nM (IC50) |
Chemical Information
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CAS No. 3032818-67-7
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Molecular Weight 688.73
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Formula C38H34F2N8O3
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SMILES
O=C1NN=C(CC2=CC=C(F)C(C(N3CCN(CC4=CC(NC5=NC=NC(C6=CC=C(F)C=C6OCC)=C5)=NC=C4)CC3)=O)=C2)C7=C1C=CC=C7
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)