3 Results for "

(-)-Bicuculline methochloride

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "(-)-Bicuculline methochloride" in MCE Product Catalog:

44
44 Publications Verification
Cat. No.: HY-137790
CAS No.: 38641-83-7
Purity:  99.35%
Synonyms: (-)-Bicuculline methochloride
Target:  

GABA Receptor

Research Areas:  

Neurological Disease

Bicuculline ((+)-Bicuculline; d-Bicuculline) methochloride is a selective GABAA receptor antagonist with an IC50 value of 3 μM. Bicuculline methochloride induces clonic tonic convulsions in mammals and can also be used to block Ca 2+ activated potassium channels. Bicuculline methochloride can be used in studies of epilepsy and other related psychiatric disorders .
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Cat. No.: HY-100783A
CAS No.: 53552-05-9
Target:  

GABA Receptor

Research Areas:  

Neurological Disease

(+)-Bicuculline methobromide is a potent GABAA blocker. (+)-Bicuculline methobromide alters membrane properties and firing pattern. (+)-Bicuculline methobromide reduces the Apamin-sensitive afterhyperpolarization, while Apamin is a toxin isolated from bee venom to block small conductance Ca 2+ -activated K + channels. (+)-Bicuculline methobromide facilitates burst firing via blocking apamin-sensitive Ca 2+ -activated K + current .
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5
5 Cited Publications
Cat. No.: HY-103474
CAS No.: 40709-69-1
Purity:  99.93%
Synonyms: (-)-Bicuculline methiodide
Target:  

GABA Receptor

Research Areas:  

Neurological Disease

Bicuculline methiodide ((-)-Bicuculline methiodide) is a potent GABAA blocker. Bicuculline methiodide alters membrane properties and firing pattern. Bicuculline methiodide reduces the Apamin-sensitive afterhyperpolarization, while Apamin is a toxin isolated from bee venom to block small conductance Ca 2+ -activated K + channels. Bicuculline methiodide facilitates burst firing via blocking apamin-sensitive Ca 2+ -activated K + current .
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