5 Results for "

(-)-Isopenbutolol

" in MedChemExpress (MCE) Product Catalog:
Products (5)

5 Results for "(-)-Isopenbutolol" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-116790
CAS No.: 38363-40-5
Synonyms: (S)-Penbutolol; (-)-Isopenbutolol
Research Areas:  

Neurological Disease

(-)-Penbutolol ((S)-Penbutolol) is a potent β-adrenoceptor and 5-HT receptor antagonist with Ki values of 11.6 nM and 11.9 nM for 5-HT in rat cornu ammonis 1 (CA1) and human CA3 .
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Cat. No.: HY-116790A
CAS No.: 38363-41-6
Purity:  ≥95.0%
Synonyms: (R)-Penbutolol; (+)-Isopenbutolol
Target:  

Adrenergic Receptor

Research Areas:  

Metabolic Disease Endocrinology

(+)-Penbutolol is a β-adrenoceptor antagonist, with an IC50 of 0.74 μM . (+)-Penbutolol is an optical isomer of l-penbutolol with Na + channel-blocking action .
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Cat. No.: HY-116790BS
CAS No.: 1346747-40-7
Synonyms: (Rac)-Penbutolol-d9; (±)-Isopenbutolol-d9
(±)-Penbutolol-d9 is the deuterium labeled (±)-Penbutolol .
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Cat. No.: HY-116790B
CAS No.: 36507-48-9
Synonyms: (Rac)-Penbutolol; (±)-Isopenbutolol
Target:  

Adrenergic Receptor

Research Areas:  

Cardiovascular Disease

(±)-Penbutolol ((Rac)-Penbutolol) is the racemic mixture of Penbutolol. (±)-Penbutolol is an orally active β-adrenergic receptor antagonist. (±)-Penbutolol antagonizes exercise-induced tachycardia, reduces the increase in peak expiratory flow rate (PEFR) caused by exercise, and decreases resting plasma renin activity (PRA). (±)-Penbutolol reaches peak plasma concentration 1 hour after oral administration, with a half-life of 4.5 hours, and is converted into an active metabolite in the body. (±)-Penbutolol can be used in cardiovascular-related disease research .
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Cat. No.: HY-116790BSA
CAS No.: 1346605-01-3
Synonyms: (Rac)-Penbutolol-d9 hydrochloride; (±)-Isopenbutolol-d9 hydrochloride
(±)-Penbutolol-d9 (hydrochloride) is a deuterium labeled (±)-Penbutolol hydrochloride. (+)-Penbutolol hydrochloride is a β-adrenoceptor antagonist, with an IC50 of 0.74 μM .
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